Exploiting Hydrophobic Amino Acid Scanning to Develop Cyclic Peptide Inhibitors of the SARS-CoV-2 Main Protease with Antiviral Activity
Katriona Harrison, Patrick W. Carlos, Sven Ullrich, Anupriya Aggarwal, Jason Johansen‐Leete, Vishnu Mini Sasi, Isabel Barter, Joshua WC. Maxwell, Max J. Bedding, Mark Larance, Stuart Turville, Alexander Norman, Colin J. Jackson, Christoph Nitsche, and Richard J. Payne*
Chemistry – A European Journal, 2024
A broad-spectrum macrocyclic peptide inhibitor of the SARS-CoV-2 spike protein
Vito Thijssen, Daniel L. Hurdiss, Oliver J. Debski-Antoniak, Matthew A. Spence, Charlotte Franck, Alexander Norman, Anupriya Aggarwal, Nadia J. Mokiem, David A.A. van Dongen, Stein W Vermeir, Minglong Liu, Wentao Li, Marianthi Chatziandreou, Tim Donselaar, Wenjuan Du, Ieva Drulyte, Berend-Jan Bosch, Joost Snijder, Stuart G. Turville, Richard J. Payne, Colin J. Jackson, Frank J.M. van Kuppeveld*, Seino A.K. Jongkees*
A broad-spectrum macrocyclic peptide inhibitor of the SARS-CoV-2 spike protein
Proceedings of the National Academy of Sciences, 2023